Pregnane X Receptor [pregnanový X receptor]

topical
25
Terms

NR1I2
pregnanový receptor X
PXR
steroid X receptor
SXR

 

NR1I2
Nuclear Receptor Subfamily 1, Group I, Member 2
Steroid and Xenobiotic Receptor
Steroid X Receptor
SXR Receptor

Definition

Steroid receptor that binds and is activated by variety of endogenous compounds and XENOBIOTICS. It binds the response element in promoters of genes that encode CYTOCHROME P450 3A4 and ATP BINDING CASSETTE TRANSPORTER, SUBFAMILY B, MEMBER 1 proteins, and also activates the transcription of multiple genes involved in the metabolism and secretion of potentially harmful xenobiotics, drugs, and endogenous compounds. It is activated by the antibiotic RIFAMPICIN and various plant metabolites, such as hyperforin, guggulipid, colupulone, and ISOFLAVONES.

DUI
D000077297 MeSH Browser
CUI
M0287170
History note
2019 (1998)
Public note
2019; PREGNANE X RECEPTOR was indexed under RECEPTORS, STEROID 2007-2018; and under RECEPTORS, CYTOPLASMIC AND NUCLEAR 1998-2006

D Chemicals and Drugs
D12.776 Proteins 2 581
D12.776.826.750 Receptors, Steroid 143
D12.776.826.750.038 Oxysterol Binding Proteins
D12.776.826.750.075 Pregnane X Receptor 25
D12.776.826.750.150 Receptors, Androgen 162
D12.776.826.750.350 Receptors, Estrogen 340
D12.776.826.750.430 Receptors, Glucocorticoid 107
D12.776.826.750.530 Receptors, Mineralocorticoid 29
D12.776.826.750.765 Receptors, Progesterone 132
D12.776.930 Transcription Factors 733
D12.776.930.778 Receptors, Steroid 143
D12.776.930.778.175 Pregnane X Receptor 25
D12.776.930.778.350 Receptors, Estrogen 340

NR1I2 protein, human Chemical MeSH Browser

Nr1i2 protein, mouse Chemical MeSH Browser

Nr1i2 protein, rat Chemical MeSH Browser