PCSK9 Inhibitors [PCSK9 inhibitory]

topical
244
Terms

inhibitory PCSK9
kardiovaskulární inhibitory PCSK9
kardiovaskulární PCSK9 inhibitory

 

PCSK9 Inhibitors Cardiovascular
PCSK9 Inhibitors, Cardiovascular

Definition

Agents that inhibit Proprotein Convertase Subtilisin/Kexin Type 9 (see PROPROTEIN CONVERTASE 9 (PCSK9)), an enzyme that plays an important role in the degradation of the LDL receptors. It favors LDL catabolism and reduces plasma LDL-cholesterol (LDL_C) level.

DUI
D000091362 MeSH Browser
CUI
M000748765
Previous indexing
Anticholesteremic Agents (2018-2021)
History note
2022
Public note
2022

D Chemicals and Drugs
D27.505.519.186 Antimetabolites 120
D27.505.519.186.071 Hypolipidemic Agents 1 627
D27.505.519.186.071.202 Anticholesteremic Agents 411
D27.505.519.186.071.202.370 Hydroxymethylglutaryl-CoA Reductase Inhibitors 1 841
D27.505.519.186.071.202.685 PCSK9 Inhibitors 244
D27.505.519.389 Enzyme Inhibitors 880
D27.505.519.389.745 Protease Inhibitors 273
D27.505.519.389.745.800 Serine Proteinase Inhibitors 49
D27.505.519.389.745.800.449 Antithrombins 252
D27.505.519.389.745.800.506 PCSK9 Inhibitors 244
D27.505.519.389.745.800.562 Serine Peptidase Inhibitors, Kazal Type
D27.505.519.389.745.800.675 Serpins 41
D27.505.519.389.745.800.900 Trypsin Inhibitors 122
D27.505.954 Therapeutic Uses 61
D27.505.954.557 Lipid Regulating Agents 8
D27.505.954.557.500 Hypolipidemic Agents 1 627
D27.505.954.557.500.202 Anticholesteremic Agents 411
D27.505.954.557.500.202.370 Hydroxymethylglutaryl-CoA Reductase Inhibitors 1 841
D27.505.954.557.500.202.685 PCSK9 Inhibitors 244