rozpřahující látky [Uncoupling Agents]

tematický
24
Termíny

odpojovače

Perzistentní odkaz   https://www.medvik.cz/link/D014475
Definice

Chemické látky, které v metabolickém cyklu oddělují oxidaci od fosforylace, takže nedochází k syntéze ATP. Patří sem ty ionofory, které narušují přenos elektronů zkratováním protonového gradientu přes mitochondriální membrány.

Chemical agents that uncouple oxidation from phosphorylation in the metabolic cycle so that ATP synthesis does not occur. Included here are those IONOPHORES that disrupt electron transfer by short-circuiting the proton gradient across mitochondrial membranes.

Anotace
enzyme inhib
DUI
D014475 MeSH Prohlížeč
CUI
M0022252
Předchozí užití
Oxidative Phosphorylation/drug effects (1966-1968); Oxidoreductases/antagonists & inhibitors (1968)
Historická pozn.
72(69)
Veřejná pozn.
72; DIO-9 was see under ANTIBIOTICS 1975-81

D Chemikálie a léčiva
D09 sacharidy 723
D10 lipidy 2 524
D27.505.519.389 inhibitory enzymů 873
D27.505.519.389.092 inhibitory adenosindeaminasy 6
D27.505.519.389.108 inhibitory adenylylcyklasy 14
D27.505.519.389.174 inhibitory kalcineurinu 122
D27.505.519.389.200 inhibitory karboanhydras 59
D27.505.519.389.275 cholinesterasové inhibitory 967
D27.505.519.389.310 inhibitory cyklooxygenasy 454
D27.505.519.389.335 inhibitory cytochromu P450 93
D27.505.519.389.350 antagonisté kyseliny listové 67
D27.505.519.389.360 inhibitory histondeacetylas 110
D27.505.519.389.370 statiny 1 837
D27.505.519.389.375 inhibitory integrasy 4
D27.505.519.389.400 inhibitory beta-laktamasy 74
D27.505.519.389.480 inhibitory lipoxygenas 51
D27.505.519.389.616 inhibitory MAO 155
D27.505.519.389.735 inhibitory fosfodiesteras 405
D27.505.519.389.737 inhibitory fosfolipasy A2 9
D27.505.519.389.739 PARP inhibitory 185
D27.505.519.389.740 inhibitory prolylhydroxylas 3
D27.505.519.389.745 inhibitory proteas 272
D27.505.519.389.755 inhibitory proteinkinas 1 364
D27.505.519.389.760 inhibitory syntézy proteinů 37
D27.505.519.389.848 inhibitory protonové pumpy 489
D27.505.519.389.870 inhibitory syntézy steroidů 1
D27.505.519.389.892 inhibitory topoisomeras 7
D27.505.519.389.936 rozpřahující látky 24
D27.505.519.389.936.500 protonové ionofory 1