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Extracellular hypotonicity induces disturbance of sodium currents in rat ventricular myocytes
L. Hu, J. Ma, P. Zhang, J. Zheng
Jazyk angličtina Země Česko
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- MeSH
- benzylaminy farmakologie MeSH
- chelátory farmakologie MeSH
- EGTA analogy a deriváty farmakologie MeSH
- financování organizované MeSH
- hypotonické roztoky MeSH
- indoly farmakologie MeSH
- inhibitory proteinkinas farmakologie MeSH
- kardiomyocyty metabolismus účinky léků MeSH
- kationtové kanály TRPV antagonisté a inhibitory metabolismus MeSH
- kinetika MeSH
- krysa rodu rattus MeSH
- maleimidy farmakologie MeSH
- membránové potenciály MeSH
- metoda terčíkového zámku MeSH
- proteinkinasa C antagonisté a inhibitory metabolismus MeSH
- proteinkinasa závislá na vápníku a kalmodulinu typ 2 antagonisté a inhibitory metabolismus MeSH
- rutheniová červeň farmakologie MeSH
- signální transdukce účinky léků MeSH
- sodík metabolismus MeSH
- srdeční komory cytologie metabolismus účinky léků MeSH
- sulfonamidy farmakologie MeSH
- vápník metabolismus MeSH
- zvířata MeSH
- Check Tag
- krysa rodu rattus MeSH
- mužské pohlaví MeSH
- ženské pohlaví MeSH
- zvířata MeSH
Hypotonic solution alters ion channel activity, but little attention has been paid to voltage-dependent sodium channels. The aim of this study was to investigate the effects of hypotonic solution on transient sodium currents (INaT) and persistent sodium currents (INaP). We also explored whether the intracellular signal transduction systems participated in the hypotonic modifications of sodium currents. INaT and INaP were recorded by means of whole-cell patch-clamp technique in isolated rat ventricular myocytes. Our results revealed that hypotonic solution reduced INaT and simultaneously augmented INaP with the occurrence of interconversion between INaT and INaP. Hypotonic solution shifted steady-state inactivation to a more negative potential, prolonged the time of recovery from inactivation, and enhanced intermediate inactivation (IIM). Ruthenium red (RR, inhibitor of TRPV4), bisindolylmaleimide VI (BIM, inhibitor of PKC), Kn-93 (inhibitor of Ca/CaMKII) and BAPTA (Ca2+-chelator) inhibited the effects of hypotonic solution on INaT and INaP. Therefore we conclude that hypotonic solution inhibits INaT, enhances INaP and IIM with the effects being reversible. TRPV4 and intracellular Ca2+, PKC and Ca/CaMKII participate in the hypotonic modifications of sodium currents.
Citace poskytuje Crossref.org
Lit.: 35
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- $a Hypotonic solution alters ion channel activity, but little attention has been paid to voltage-dependent sodium channels. The aim of this study was to investigate the effects of hypotonic solution on transient sodium currents (INaT) and persistent sodium currents (INaP). We also explored whether the intracellular signal transduction systems participated in the hypotonic modifications of sodium currents. INaT and INaP were recorded by means of whole-cell patch-clamp technique in isolated rat ventricular myocytes. Our results revealed that hypotonic solution reduced INaT and simultaneously augmented INaP with the occurrence of interconversion between INaT and INaP. Hypotonic solution shifted steady-state inactivation to a more negative potential, prolonged the time of recovery from inactivation, and enhanced intermediate inactivation (IIM). Ruthenium red (RR, inhibitor of TRPV4), bisindolylmaleimide VI (BIM, inhibitor of PKC), Kn-93 (inhibitor of Ca/CaMKII) and BAPTA (Ca2+-chelator) inhibited the effects of hypotonic solution on INaT and INaP. Therefore we conclude that hypotonic solution inhibits INaT, enhances INaP and IIM with the effects being reversible. TRPV4 and intracellular Ca2+, PKC and Ca/CaMKII participate in the hypotonic modifications of sodium currents.
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