Disintegrins [disintegriny]
- Terms
-
Disintegrin
A family of polypeptides purified from snake venoms, which contain the arginine-glycine-aspartic acid (RGD) sequence. The RGD tripeptide binds to integrin receptors and thus competitively inhibits normal integrin-ligand interactions. Disintegrins thus block adhesive functions and act as platelet aggregation inhibitors.
- Annotation
- polypeptides from snake venom; platelet aggregation inhib
- polypeptidy z hadího jedu; inhibitor agregace krevních destiček
- DUI
- D019483 MeSH Browser
- CUI
- M0028974
- Previous indexing
- Peptides (1992-1996); Venoms (1992-1994)
- History note
- 97; was DISINTEGRINS (NM) 1992-96
- Online note
- use DISINTEGRINS (NM) to search DISINTEGRINS 1992-96
- Public note
- 97; DISINTEGRINS was indexed under PEPTIDES 1992-96 & VENOMS 1992-94
Allowable subheadings
- AD
- administration & dosage
- AE
- adverse effects
- AG
- agonists
- AN
- analysis
- AI
- antagonists & inhibitors
- BI
- biosynthesis
- BL
- blood
- CF
- cerebrospinal fluid
- CS
- chemical synthesis
- CH
- chemistry
- CL
- classification
- DF
- deficiency
- DE
- drug effects
- EC
- economics
- GE
- genetics
- HI
- history
- IM
- immunology
- IP
- isolation & purification
- ME
- metabolism
- PK
- pharmacokinetics
- PD
- pharmacology
- PH
- physiology
- PO
- poisoning
- RE
- radiation effects
- ST
- standards
- SD
- supply & distribution
- TU
- therapeutic use
- TO
- toxicity
- UR
- urine
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