Multidrug Resistance-Associated Proteins [proteiny spojené s mnohočetnou rezistencí k lékům]
- Terms
-
ATP-Binding Cassette, Sub-Family C Proteins
MOAT Protein
Multidrug Resistance-Associated Protein
Multispecific Organic Anion Transport Proteins
Multispecific Organic Anion Transporter
A sequence-related subfamily of ATP-BINDING CASSETTE TRANSPORTERS that actively transport organic substrates. Although considered organic anion transporters, a subset of proteins in this family have also been shown to convey drug resistance to neutral organic drugs. Their cellular function may have clinical significance for CHEMOTHERAPY in that they transport a variety of ANTINEOPLASTIC AGENTS. Overexpression of proteins in this class by NEOPLASMS is considered a possible mechanism in the development of multidrug resistance (DRUG RESISTANCE, MULTIPLE). Although similar in function to P-GLYCOPROTEINS, the proteins in this class share little sequence homology to the ATP BINDING CASSETTE TRANSPORTER, SUBFAMILY B, MEMBER 1 family of proteins.
- DUI
- D027425 MeSH Browser
- CUI
- M0238823
- Previous indexing
- P-Glycoprotein (1987-2001)
- History note
- 2002; use MULTIDRUG RESISTANCE-ASSOCIATED PROTEINS (NM) 1994-2001; for MOAT PROTEIN & MULTISPECIFIC ORGANIC ANION TRANSPORTER use ANION TRANSPORT PROTEINS 1995-2001
- Public note
- 2002; MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN was indexed under ABC TRANSPORTERS 1994-2001; MOAT PROTEIN & MULTISPECIFIC ORGANIC ANION TRANSPORTER were indexed under CARRIER PROTEINS 1995-2001
Allowable subheadings
- AD
- administration & dosage
- AE
- adverse effects
- AG
- agonists
- AN
- analysis 14
- AI
- antagonists & inhibitors 3
- BI
- biosynthesis 3
- BL
- blood 1
- CF
- cerebrospinal fluid
- CS
- chemical synthesis
- CH
- chemistry 2
- CL
- classification
- DF
- deficiency
- DE
- drug effects 2
- EC
- economics
- GE
- genetics 27
- HI
- history
- IM
- immunology 3
- IP
- isolation & purification 1
- ME
- metabolism 34
- PK
- pharmacokinetics 1
- PD
- pharmacology
- PH
- physiology 4
- PO
- poisoning
- RE
- radiation effects
- ST
- standards
- SD
- supply & distribution
- TU
- therapeutic use
- TO
- toxicity
- UL
- ultrastructure
- UR
- urine
ABCC10 protein, human Chemical MeSH Browser
ABCC4 protein, human Chemical MeSH Browser
ABCC5 protein, human Chemical MeSH Browser
ABCC5 protein, zebrafish Chemical MeSH Browser
ABCC6 protein, human Chemical MeSH Browser
ATMRP5 protein, Arabidopsis Chemical MeSH Browser
Abcc10 protein, mouse Chemical MeSH Browser
Abcc4 protein, mouse Chemical MeSH Browser
Abcc4 protein, rat Chemical MeSH Browser
Abcc4 protein, zebrafish Chemical MeSH Browser
Abcc5 protein, mouse Chemical MeSH Browser
Abcc5 protein, rat Chemical MeSH Browser
Abcc6 protein, mouse Chemical MeSH Browser
Abcc6 protein, rat Chemical MeSH Browser
AcrB protein, E coli Chemical MeSH Browser
BaeR protein, Salmonella typhimurium Chemical MeSH Browser
BaeS protein, Salmonella typhimurium Chemical MeSH Browser
CDR-2 protein, Candida albicans Chemical MeSH Browser
DrrA protein, Streptomyces peucetius Chemical MeSH Browser
DrrB protein, Streptomyces peucetius Chemical MeSH Browser
HV126 protein, human Chemical MeSH Browser
LmrA protein, Lactococcus lactis Chemical MeSH Browser
LmrC protein, Lactococcus lactis Chemical MeSH Browser
LmrD protein, Lactococcus lactis Chemical MeSH Browser
MRP-4 protein, C elegans Chemical MeSH Browser
MRP4 protein, Drosophila Chemical MeSH Browser
MRP6 protein, Arabidopsis Chemical MeSH Browser
Mdr1 protein, Plasmodium falciparum Chemical MeSH Browser
Mdr1 protein, Plasmodium vivax Chemical MeSH Browser
Mdr2 protein, Plasmodium falciparum Chemical MeSH Browser
NorA protein, Staphylococcus Chemical MeSH Browser
RamA protein, Salmonella typhimurium Chemical MeSH Browser
RamR protein, Salmonella typhimurium Chemical MeSH Browser
Slco2b1 protein, rat Chemical MeSH Browser
TolC protein, Legionella pneumophila Chemical MeSH Browser
mrp-7 protein, C elegans Chemical MeSH Browser
multi-resistance associated protein 1, zebrafish Chemical MeSH Browser
multidrug resistance transporter STY2458, Salmonella typhi Chemical MeSH Browser
multidrug resistance-associated protein 1 Chemical MeSH Browser
multidrug resistance-associated protein 3 Chemical MeSH Browser