inhibitory dipeptidylpeptidasy 4 [Dipeptidyl-Peptidase IV Inhibitors]

tematický
572
Termíny

dipeptidylpeptidasa IV - inhibitory
DPP-4 inhibitory
gliptiny
inhibitory dipeptidylpeptidázy 4
inhibitory DPP-4

 

Dipeptidyl Peptidase 4 Inhibitor
Dipeptidyl-Peptidase 4 Inhibitor
Dipeptidyl-Peptidase 4 Inhibitors
Dipeptidyl-Peptidase IV Inhibitor
DPP-4 Inhibitor
DPP-4 Inhibitors
DPP-IV Inhibitor
DPP-IV Inhibitors
DPP4 Inhibitor
DPP4 Inhibitors
Gliptin
Gliptins

Perzistentní odkaz   https://www.medvik.cz/link/D054873
Definice

Sloučeniny, které potlačují degradaci inkretinů blokováním účinku dipeptidylpeptidázy 4. To pomáhá korigovat defektní sekreci insulinu a glukagonu charakteristickou pro diabetes mellitus 2. typu tím, že stimuluje sekreci inzulinu a potlačuje uvolňování glukagonu.

Compounds that suppress the degradation of INCRETINS by blocking the action of DIPEPTIDYL-PEPTIDASE IV. This helps to correct the defective INSULIN and GLUCAGON secretion characteristic of TYPE 2 DIABETES MELLITUS by stimulating insulin secretion and suppressing glucagon release.

DUI
D054873 MeSH Prohlížeč
CUI
M0508515
Historická pozn.
2008
Veřejná pozn.
2008

D Chemikálie a léčiva
D27.505.519.389 inhibitory enzymů 873
D27.505.519.389.745 inhibitory proteas 272
D27.505.519.389.745.085 inhibitory ACE 2 038
D27.505.519.389.745.325 inhibitory cysteinových proteinas 30
D27.505.519.389.745.335 inhibitory dipeptidylpeptidasy 4 572
D27.505.519.389.745.705 inhibitory proteasomu 95
D27.505.519.389.745.753 inhibitory reninu
D27.505.519.389.745.800 inhibitory serinových proteinas 49
D27.505.519.389.745.900 inhibitory virových proteáz 6
D27.505.696.422 hypoglykemika 2 719
D27.505.696.422.500 inhibitory dipeptidylpeptidasy 4 572
D27.505.696.422.625 sekretagoga insulinu
D27.505.696.422.688 agonisté PPAR gama
D27.505.696.422.750 glifloziny 780