Direct C-H borylation and C-H arylation of pyrrolo[2,3-d]pyrimidines: synthesis of 6,8-disubstituted 7-deazapurines
Language English Country Great Britain, England Media print-electronic
Document type Journal Article, Research Support, Non-U.S. Gov't
PubMed
19225668
DOI
10.1039/b900218a
Knihovny.cz E-resources
- MeSH
- Catalysis MeSH
- Purines chemical synthesis MeSH
- Pyrimidines chemistry MeSH
- Pyrroles chemistry MeSH
- Boron Compounds chemistry MeSH
- Tubercidin MeSH
- Publication type
- Journal Article MeSH
- Research Support, Non-U.S. Gov't MeSH
- Names of Substances
- Purines MeSH
- Pyrimidines MeSH
- Pyrroles MeSH
- Boron Compounds MeSH
- Tubercidin MeSH
Novel direct C-H borylations of 7-deazapurines to position 8 by B2pin2 under Ir catalysis were followed by Suzuki cross-couplings with aryl halides and other functional group transformations to give diverse 8-substituted 7-deazaadenines.
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