Hirudins [hirudiny]
- Terms
-
hirudin
-
Hirudin
Single-chain polypeptides of about 65 amino acids (7 kDa) from LEECHES that have a neutral hydrophobic N terminus, an acidic hydrophilic C terminus, and a compact, hydrophobic core region. Recombinant hirudins lack tyr-63 sulfation and are referred to as 'desulfato-hirudins'. They form a stable non-covalent complex with ALPHA-THROMBIN, thereby abolishing its ability to cleave FIBRINOGEN.
- DUI
- D006629 MeSH Browser
- CUI
- M0465835
- History note
- 2005(1963)
- Public note
- 2005; see HIRUDIN 1963-2004
Combination
- therapeutic use
- Hirudin Therapy
Allowable subheadings
- AD
- administration & dosage 9
- AE
- adverse effects 3
- AG
- agonists
- AN
- analysis
- AI
- antagonists & inhibitors 1
- BI
- biosynthesis
- BL
- blood 1
- CF
- cerebrospinal fluid
- CS
- chemical synthesis
- CH
- chemistry 1
- CL
- classification 1
- DE
- drug effects
- EC
- economics
- GE
- genetics
- HI
- history
- IM
- immunology
- IP
- isolation & purification
- ME
- metabolism 1
- PK
- pharmacokinetics
- PD
- pharmacology 7
- PH
- physiology 1
- PO
- poisoning
- RE
- radiation effects
- ST
- standards
- SD
- supply & distribution
- TO
- toxicity
- UL
- ultrastructure
- UR
- urine
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