In vitro antibacterial and antifungal activity of salicylanilide benzoates
Jazyk angličtina Země Spojené státy americké Médium print-electronic
Typ dokumentu časopisecké články, práce podpořená grantem
PubMed
22666101
PubMed Central
PMC3361159
DOI
10.1100/2012/290628
Knihovny.cz E-zdroje
- MeSH
- antibakteriální látky farmakologie MeSH
- antifungální látky farmakologie MeSH
- benzoáty farmakologie MeSH
- magnetická rezonanční spektroskopie MeSH
- mikrobiální testy citlivosti MeSH
- salicylanilidy farmakologie MeSH
- spektrofotometrie infračervená MeSH
- techniky in vitro MeSH
- Publikační typ
- časopisecké články MeSH
- práce podpořená grantem MeSH
- Názvy látek
- antibakteriální látky MeSH
- antifungální látky MeSH
- benzoáty MeSH
- salicylanilide MeSH Prohlížeč
- salicylanilidy MeSH
The resistance to antimicrobial agents brings a need of novel antimicrobial agents. We have synthesized and found the in vitro antibacterial activity of salicylanilide esters with benzoic acid (2-(phenylcarbamoyl)phenyl benzoates) in micromolar range. They were evaluated in vitro for the activity against eight fungal and eight bacterial species. All derivatives showed a significant antibacterial activity against Gram-positive strains with minimum inhibitory concentrations ≥ 0.98 μmol/L including methicillin-resistant Staphylococcus aureus strain. The most active compounds were 5-chloro-2-(3,4-dichlorophenylcarbamoyl)phenyl benzoate and 4-chloro-2-(4-(trifluoromethyl)phenylcarbamoyl)phenyl benzoate. The antifungal activity is significantly lower.
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